Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,216
Tocris Bioscience™ (RS)-MCPG
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CAS: 146669-29-6 Molecular Formula: C10H11NO4
| CAS | 146669-29-6 |
|---|---|
| Molecular Formula | C10H11NO4 |
1,217
Tocris Bioscience™ Diphenhydramine hydrochloride
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CAS: 147-24-0 Molecular Formula: C17H22ClNO
| CAS | 147-24-0 |
|---|---|
| Molecular Formula | C17H22ClNO |
1,218
Tocris Bioscience™ CC4
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High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist
| Target | Additional Nicotinic (a4b2) Receptor Compounds |
|---|---|
| CAS | 492-02-4 |
| Purity | >98% |
| Chemical Name or Material | (1R,5S)-1,2,3,4,5,6-Hexahydro-3-[2-[(1R,5S)-1,5,6,8-tetrahydro-8-oxo-1,5-methano-2H-pyrido[1,2-a][1,5]diazocin-3(4H)-yl]ethyl]-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C24H30N4O2 |
| Formula Weight | 406.52 |
1,219
Tocris Bioscience™ TFB-TBOA
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High affinity EAAT1 and EAAT2 blocker
| CAS | 480439-73-4 |
|---|---|
| Solubility | Soluble to 100mM in DMSO |
| Chemical Name or Material | (3S)-3-[[3-[[4-(Trifluoromethyl)benzoyl]amino]phenyl]methoxy]-L-aspartic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H17F3N2O6 |
| Formula Weight | Observed MW: 426.35 |
| Assay Percent Range | >98% |
1,220
Tocris Bioscience™ TP 472
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Potent BRD9/7 inhibitor
1,221
Tocris Bioscience™ VH 032 amide-alkylC4-amine
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PROTACs (Proteolysis Targeting Chimeras)
1,222
Tocris Bioscience™ Brequinar sodium
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Potent and selective DHODH inhibitor.
| Target | DHODH Inhibitors |
|---|---|
| CAS | 96201-88-6 |
| Chemical Name or Material | 6-Fluoro-2-(2′-fluoro[1,1′-biphenyl]-4-yl)-3-methyl-4-quinolinecarboxylic acid sodium |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C23H14F2NO2Na |
| Formula Weight | Observed MW: 397.35 |
| Assay Percent Range | >99% |
1,223
Tocris Bioscience™ TP 064
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Potent and selective PRMT 4 inhibitor
| Product Type | Bioactive Small Molecule |
|---|---|
| Color | White |
| Solubility | Soluble to 100mM in 1eq. HCl and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | TP 064 |
| Recommended Storage | Store at -20°C |
| Synonym | N-Methyl-N-((2-(1-(2-(methylamino)ethyl)piperidin-4-yl)pyridin-4-yl)methyl)-3-phenoxybenzamide |
| Molecular Formula | C28H34N4O2 |
| Formula Weight | 458.6 |
1,224
Tocris Bioscience™ Bepridil hydrochloride
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CAS: 68099-86-5 Molecular Formula: C24H35ClN2O
| CAS | 68099-86-5 |
|---|---|
| Molecular Formula | C24H35ClN2O |
1,225
Tocris Bioscience™ BMS 303141
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CAS: 943962-47-8 Molecular Formula: C19H15Cl2NO4S
| CAS | 943962-47-8 |
|---|---|
| Molecular Formula | C19H15Cl2NO4S |
1,226
Tocris Bioscience™ CFTRinh 172
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CAS: 307510-92-5 Molecular Formula: C18H10F3NO3S2
| CAS | 307510-92-5 |
|---|---|
| Molecular Formula | C18H10F3NO3S2 |
1,227
Tocris Bioscience™ Lovastatin
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CAS: 75330-75-5 Molecular Formula: C24H36O5
| CAS | 75330-75-5 |
|---|---|
| Molecular Formula | C24H36O5 |
1,228
Tocris Bioscience™ W 54011
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High affinity C5a receptor antagonist
| Target | Complement Signaling inhibitors |
|---|---|
| CAS | 405098-33-1 |
| Purity | >98% |
| Chemical Name or Material | N-[[4-(Dimethylamino)phenyl]methyl]-1,2,3,4-tetrahydro-7-methoxy-N-[4-(1-methylethyl)phenyl]-1-naphthalenecarboxamide hydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C30H36N2O2.HCl |
| Formula Weight | 493.08 |
1,229
Tocris Bioscience™ NBI 27914 hydrochloride
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CAS: 1215766-76-9 Molecular Formula: C18H21Cl5N4
| CAS | 1215766-76-9 |
|---|---|
| Molecular Formula | C18H21Cl5N4 |
1,230
Tocris Bioscience™ AdipoRon hydrochloride
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CAS: 1781835-20-8 Molecular Formula: C27H29ClN2O3
| CAS | 1781835-20-8 |
|---|---|
| Molecular Formula | C27H29ClN2O3 |